TargetMol

EP300/CBP ligand 2

Product Code:
 
TAR-T89972
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20°C
 

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Further Information

Bioactivity:
EP300/CBP ligand 2 (compound S19) serves as a specific ligand for the bromodomain of CREB binding protein (CBP) and E1A-associated protein (EP300). It plays a critical role in PROTAC technology by acting as a target protein ligand. By linking to an E3 ubiquitin ligase ligand via the PROTAC Linker, it facilitates the synthesis of PROTAC molecules capable of targeted protein degradation. For instance, when EP300/CBP ligand 2 is connected to the conjugate (E3 ubiquitin enzyme ligand + Linker) Thalidomide-NH-C10-Boc, it results in the formation of the PROTAC molecule dCE-2.
Formula:
C20H18N6O
Molecular Weight:
358.4
Pathway:
Chromatin/Epigenetic; PROTAC
Purity:
98%
Target:
Epigenetic Reader Domain; Ligands for Target Protein for PROTAC

Documents